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Vapitadine dihydrochloride
🥰Excellent
Catalog No. T29096Cas No. 279253-83-7
Alias Vapitadine 2HCl, R-129160 dihydrochloride, R129160 dihydrochloride, R-129160 2HCl, R129160 2HCl, R 129160 2HCl
Vapitadine dihydrochloride(R-129160 2HCl) is a novel, potent, selective and non-sedating compound with inhibitory effects on histamine H1.
Vapitadine dihydrochloride
🥰Excellent
Purity: 100%
Catalog No. T29096Alias Vapitadine 2HCl, R-129160 dihydrochloride, R129160 dihydrochloride, R-129160 2HCl, R129160 2HCl, R 129160 2HClCas No. 279253-83-7
Vapitadine dihydrochloride(R-129160 2HCl) is a novel, potent, selective and non-sedating compound with inhibitory effects on histamine H1.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $258 | In Stock | |
| 5 mg | $642 | In Stock | |
| 10 mg | $913 | In Stock | |
| 25 mg | $1,370 | In Stock | |
| 50 mg | $1,850 | In Stock |
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Purity:100%
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | Vapitadine dihydrochloride(R-129160 2HCl) is a novel, potent, selective and non-sedating compound with inhibitory effects on histamine H1. |
| Alias | Vapitadine 2HCl, R-129160 dihydrochloride, R129160 dihydrochloride, R-129160 2HCl, R129160 2HCl, R 129160 2HCl |
| Molecular Weight | 369.29 |
| Formula | C17H22Cl2N4O |
| Cas No. | 279253-83-7 |
| Smiles | O=C(C1=CN=C2N1CCC3=C(C24CCNCC4)C=CC=C3)N.Cl.Cl |
| Relative Density. | no data available |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
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DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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